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In contrast to drugs acting from the outside on cell membrane constituents, agents acting in the cell’s interior need to penetrate the cell membrane. The cell membrane basically consists of a phospholipid bilayer (80A = 8 nm in thickness) in which are embedded proteins (integral membrane proteins, such as receptors and transport molecules).
In cardiac arrest epinephrine can be used to reinitiate heart beat. Sinus tachycardia (resting rate >100 beats/min). ?-Blockers eliminate sympathoexcitation and decrease cardiac rate. Atrial flutter or fibrillation. An excessive ventricular rate can be decreased by verapamil or cardiac glycosides. |
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