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Chloroquine and quinine accumulate within the acidic vacuoles of blood schizonts and inhibit polymerization of heme, the latter substance being toxic for the schizonts. Antimalarial drug choice takes into account tolerability and plasmodial resistance. Tolerability. The first available antimalarial, quinine, has the smallest therapeutic margin.
Since they may cause mucosal damage, their use should be short-term. |
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