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With oral administration, dividing the total daily dose into several individual ones, e. g. , four, three, or two, offers a practical compromise. When the daily dose is given in several divided doses, the mean plasma level shows little fluctuation. In practice, it is found that a regimen of frequent regular drug ingestion is not well adhered to by patients.
Hepatic elimination obeys exponential kinetics because metabolizing enzymes operate in the quasilinear region of their concentration-activity curve; hence the amount of drug metabolized per unit of time diminishes with decreasing blood concentration. |
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